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β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Cusbo CAS:24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Cusbowaa coenzyme oo si weyn ugu baahsan walxaha nool, Ka qaybqaata falgallada yaraynta oksaydhka. Waxay u adeegtaa sidii side elektaroonig ah oo ku jira tiro falcelin ah, iyadoo si kale loo oksaydheeyay (NADP+) iyo la dhimay (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Cusbowaa walax ay nicotinic acid amide adenine dinucleotide iyo molecule fosfate ku xiran yihiin xiriirka ester. Waa soo-dhoweeye haydarojiin ah waxaana loo isticmaali karaa horumarinta iyo horumarinta noocyo kala duwan oo ah falgalayaasha ogaanshaha in vitro.
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β-Nicotinamide Adenine Dinucleotide Lithium cusbo (NAD Lithium cusbo) CAS: 64417-72-7
β-Nicotinamide Adenine Dinucleotide Lithium cusbowaa coenzyme xudunta u ah dheef-shiid kiimikaadka. NAD oo laga helo dhammaan unugyada nool, waxaa loogu yeeraa dinucleotide sababtoo ah waxay ka kooban tahay laba nucleotide oo ku biiray kooxahooda fosfate. Hal nucleotide wuxuu ka kooban yahay adenine nucleobase iyo nicotinamide kan kale. NAD wuxuu u jiraa laba qaab: qaab oksaydhaysan iyo mid la dhimay, oo loo soo gaabiyo NAD+ iyo NADH (H ee hydrogen), siday u kala horreeyaan.
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Venlafaxine CAS:93413-69-5
Venlafaxine waa daawo niyad-jabka ka hortagta oo ka mid ah fasalka serotonin iyo norepinephrine reuptake inhibitor (SNRI). Daawadan waxaa markii ugu horreysay soo saaray Wyeth gudaha 19Chemicalbook93 waxaana hadda suuq geynaya Pfizer. Daawadan waxaa loo oggolaaday daaweynta xanuunka niyad-jabka weyn (MDD), xanuunka welwelka guud (GAD), iyo niyad-jabka la xiriira walwalka.
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Ciclopirox Ethanolamine CAS:41621-49-2 Alaab-qeybiye Soo-saare
Ciclopirox ethanolamine waa wakiil ballaaran oo ka hortagga fangaska, waxay sidoo kale muujisaa firfircooni bakteeriyada ka hortagta bakteeriyada badan ee Gram-positive iyo Gram-negative, waxayna leedahay sifooyin ka hortagga bararka. Waxaa loo isticmaalaa daawaynta maqaarka ee fangaska iyo caabuqyada ciddiyaha.
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Desvenlafaxine Succinate CAS:386750-22-7
Desvenlafaxine Succinate waa dawo laba-geesood ah oo serotonin iyo norepinephrine reuptake inhibitor (SNRI) oo loo oggolaaday daaweynta xanuunka niyad-jabka weyn (MDD) ee Mareykanka sannadkii 2008. Si loo horumariyo waxtarka iyo astaanta badbaadada ee venlafaxine, Wyeth wuxuu ogaaday oo sameeyay mid ka mid ah metabolites-ka ugu waaweyn ee venlafaxine, kaas oo ah metabolite-ka O-desmethyl (desvenlafaxine).
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Doxazosin Mesylate CAS:77883-43-3 Alaab-qeybiye Soo-saare
Doxazosin mesylate waa isku-darka quinazoline kaas oo ah daawooyin door ah oo ka hortaga nooca alpha1 ee alpha adrenergic receptors. Doxazosin mesylate waa jiil cusub oo ah xannibaadaha quinazolone α1 receptor blockers oo ay samaysay shirkadda Pfizer (Mareykanka), Waxay leedahay cimri dheer, iyadoo saameyn ku leh ballaarinta xididdada dhiigga, yaraynta iska caabbinta xididdada dhiigga iyo yaraynta cadaadiska dhiigga iyada oo xannibaysa receptor a 1. Waxaa lagu taliyay dibadda inay tahay daawooyinka ugu horreeya ee kiliinikada ee ka hortagga dhiigkarka iyo daaweynta cudurka qanjirka 'prostate'.
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L-Isoleucine CAS:73-32-5 Alaab-qeybiye Soo-saare
L-Isoleucine, oo sidoo kale loo yaqaan Isoleucine, waa amino acid oo ah isomer leucine ah. Waxay muhiim u tahay isku-darka hemoglobin-ka iyo nidaaminta heerarka sonkorta dhiigga iyo tamarta. L-Isoleucine waa isomer L-leucine waana amino acid muhiim ah. Waxaa laga sameeyay threonine waana amino acid hydrophobic silsilad laan ah.
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Captopril CAS:62571-86-2 Alaab-qeybiye Soo-saare
Captopril waa daawada ugu badan ee ka hortagta enzyme-ka beddela angiotensin ee loo soo jeediyay inay tahay daawo ka hortagta dhiigkarka. Waxay xannibtaa enzyme-ka beddela angiotensin, kaas oo joojiya sameynta angiotensin II isla markaana yareeya saameynta vasoconstriction ee xididdada halbowlaha iyo xididdada dhiigga. Guud ahaan xiisadda xididdada dhiigga ayaa yaraata, taasoo keenta hoos u dhaca cadaadiska halbowlaha.
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Candesartan CAS:139481-59-7 Alaab-qeybiye Soo-saare
Candesartan waa lid-ka-hortagga soo-dhoweeyaha angiotensin II (AT1), IC50s=1.12 iyo 2.86 nM ee kiliyaha adrenal ee lo'da iyo aorta bakaylaha siday u kala horreeyaan. Si gaar ah ayuu u joojiyaa foosha uu keeno angiotensin II ee xarigyada aorta bakaylaha iyada oo aan wax saameyn ah ku yeelan foosha ay kiciyaan wakiilada kale sida norepinephrine, KCl, serotonin, PGF2α ama endothelin.
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Candesartana Cilexetila CAS:145040-37-5
Candesartan Celexetil waa ester analog ah oo ka mid ah anti-angiotensin II Candesartan (sc-217825). Ka soo horjeedka receptor-kan wuxuu ka hortagayaa isku xidhka angiotensin II, oo ah vasoconstrictor xooggan. Tani waxay leedahay saameynta guud ee vasodilation iyo mugga dhiigga ee xididada dhiigga oo kordha. Candesartan Celexetil Ester waa joojiye AT1.
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Bupropion CAS:34911-55-2 Alaab-qeybiye Soo-saare
Bupropion waa ketone aromatic ah oo ah propiophenone oo sita koox tert-butylamino ah booska 2 iyo chloro beddelka booska 3 ee giraanta phenyl. Waxay leedahay door ah sida daawada niyad-jabka, sunta deegaanka iyo xenobiotic. Waa isku-darka amino labaad, xubin ka ah monochlorobenzenes iyo ketone aromatic ah.
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Bezafibrate CAS:41859-67-0 Bixiyaha Soo-saaraha
Bezafibrate waa monocarboxylic acid amide oo laga helo isku-darka rasmiga ah ee kooxda karboksiyada ee 4-chlorobenzoic acid oo leh kooxda amino ee 2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic acid. Benafibrate waxaa loo isticmaalaa daaweynta hyperlipidaemia. Waxay leedahay door sida xenobiotic, wasakheeyaha deegaanka, geroprotector iyo daawo ka hortagta lipoemic. Waa monocarboxylic acid, aromatic ether, xubin ka mid ah monochlorobenzenes iyo monocarboxylic acid amide. Waxay si shaqo leh ula xiriirtaa propionic acid.
