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Badeecadaha

Letrozole CAS:112809-51-5 Alaab-qeybiye Soo-saare

Letrozole waa qayb ka mid ah jiilka cusub ee daawooyinka ka hortagga aromatase ee aadka loo xushay waana nooc ka mid ah benzotriazole oo si macmal ah loo sameeyay. Letrozole wuxuu joojiyaa aromatase si uu u yareeyo heerarka estrogen-ka, sidaas darteed wuxuu ka hortagaa estrogen-ka inuu kiciyo koritaanka burooyinka. Hawlgalkeeda gudaha jirka waa 150-250 jeer ka xoog badan kan jiilka koowaad ee daawada ka hortagga aromatase Amarante. Maadaama ay aad u xulan tahay, saameyn kuma yeelan doonto glucocorticoid, mineralocorticoid iyo shaqooyinka qanjirka thyroid; xitaa marka la qaato qiyaaso badan, ma yeelan doonto wax saameyn ah oo ka hortagta dheecaanka corticosteroid-ka adrenal, taasoo siinaysa tusmada daaweynta sare.


Faahfaahinta Badeecada

Calaamadaha Alaabta

Codsiga iyo Saamaynta

Letrazole waxaa lagu samayn karaa laba tallaabo laga bilaabo 4-bromomethyl-benzonitrile oo leh 1,2,4-triazole waana jiilka saddexaad ee ka hortagga aromatase. Waa joojiye aad u gaar ah oo P450arom ah kaas oo ka hortagaya in androstenedione loo beddelo estrone. Yaraynta estrogen-ka plasma-ga ayaa si degdeg ah u socotay oo muddo dheer socotay. Tan waxaa lagu gaaraa iyada oo aan la joojin biosynthesis-ka kale ee steroid-ka taasoo ka dhigaysa daawada ugu xulashada badan ee la tijaabiyay ee aromatase. Letrazole waxay leedahay firfircooni ka hortagta burooyinka, si fiican ayaa loo dulqaataa mana laha waxyeellooyin sun ah. Waa 10,000 jeer ka awood badan aminoglutethimide, in vivo, oo ah daawada ugu horreysa ee si fiican loo aasaasay ee ka hortagga aromatase.

Muunadda Badeecada

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Baakaynta Alaabta:

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Macluumaad Dheeraad ah:

Halabuurka C17H11N5
Baaritaan 99%
Muuqaalka Budada cad
Lambarka CAS. 112809-51-5
Baakad 25KG
Muddada Khafiska 2 sano
Kaydinta Ku kaydi meel qabow oo qalalan
Shahaadada ISO.

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