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Pristinamycin CAS:270076-60-3
Pristinamycin waa daawo isku dhafan oo antibiyootiko ah oo ka kooban laba qaybood oo firfircoon, pristinamycin I iyo pristinamycin II. Waxay ka tirsan tahay kooxda antibiyootikada ee streptogramin waxayna muujisaa hawlo bacteriostatic iyo bakteeriya dila oo ka dhan ah noocyo kala duwan oo bakteeriya gram-positive ah, oo ay ku jiraan Staphylococcus aureus iyo Streptococcus pneumoniae. Pristinamycin waxay u shaqeysaa iyadoo joojinaysa isku-darka borotiinka bakteeriyada, taasoo ka dhigaysa mid wax ku ool ah daaweynta caabuqyada maqaarka iyo unugyada jilicsan, caabuqyada neef-mareenka, iyo caabuqyada kale ee bakteeriyada ee ay keenaan noolaha nugul.
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Ribostamycin sulfate CAS:53797-35-6
Ribostamycin sulfate waa antibiyootig aminoglycoside ah oo laga soo qaatay Streptomyces griseoluteus. Waxay muujisaa firfircooni bakteeriya oo xooggan oo ka dhan ah noocyo badan oo bakteeriya ah oo gram-negative ah iyo qaar ka mid ah gram-positive ah iyadoo joojinaysa isku-darka borotiinka. Ribostamycin sulfate waxaa badanaa loo isticmaalaa daaweynta caabuqyada kala duwan, oo ay ku jiraan caabuqyada kaadi mareenka, caabuqyada neef-mareenka, caabuqyada maqaarka iyo unugyada jilicsan, iyo septicemia oo ay sababaan noocyada bakteeriyada ee u nugul.
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Rifampicin CAS:13292-46-1
Rifampicin, oo sidoo kale loo yaqaan rifampin, waa daawo antibiyootiko oo ballaaran oo ka tirsan kooxda rifamycin. Waxaa si weyn loogu isticmaalaa daaweynta qaaxada, baraska, iyo caabuqyada kale ee bakteeriyada. Rifampicin wuxuu u shaqeeyaa isagoo joojinaya isku-darka RNA ee bakteeriyada, taasoo carqaladeynaysa awooddooda ay ku tarmaan oo ay ku noolaadaan. Sababtoo ah firfircoonideeda xooggan ee ka hortagga jeermiska iyo waxtarka ay u leedahay noocyada bakteeriyada mycobacteria, rifampicin waa qayb muhiim ah oo ka mid ah hababka daaweynta isku dhafan ee qaaxada iyo cudurrada kale ee faafa.
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Puromycin dihydrochloride CAS:58-58-2
Puromycin dihydrochloride waa daawo awood leh oo ka hortagta antibiyootiga iyo isku-darka borotiinka oo laga soo qaatay Streptomyces alboniger. Waxaa badanaa loo isticmaalaa cilmi-baarista bayoolajiga molecular-ka si loo xakameeyo isku-darka borotiinka ee unugyada iyadoo si degdeg ah loo joojiyo turjumaadda inta lagu jiro isku-darka borotiinka. Puromycin dihydrochloride waxaa lagu daraa silsiladaha peptide-ka ee cusub, taasoo horseedaysa sii deynta polypeptides aan dhammaystirnayn iyo ugu dambeyntii dhimashada unugyada. Sababtoo ah habka gaarka ah ee ficilkiisa, puromycin dihydrochloride waa qalab qiimo leh oo lagu barto isku-darka borotiinka, shaqada ribosome, muujinta hidda-wadaha, iyo jiritaanka unugyada goobaha tijaabada.
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Protionamide CAS:14222-60-7
Protionamide waa daawo antibiyootiko ah oo ka tirsan kooxda thioamide, oo inta badan loo isticmaalo daaweynta qaaxada u adkeysata daawooyinka badan. Waxay ka shaqeysaa joojinta isku-darka aashitada mycolic ee derbiga unugyada bakteeriyada, taasoo horseedaysa burburka qaaxada Mycobacterium. Protionamide waxaa badanaa loo qoraa iyadoo lala kaashanayo daawooyinka kale ee ka hortagga qaaxada iyadoo qayb ka ah daaweyn dhammaystiran oo loogu talagalay noocyada qaaxada ee u adkeysata daawada.
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Potassium clavulanate CAS: 61177-45-5
Potassium clavulanate waa daawo β-lactamase ah oo inta badan lagu daro antibiyootiko gaar ah si kor loogu qaado waxtarkooda ka dhanka ah caabuqyada bakteeriyada. Waxay ka shaqeysaa ka hortagga burburka antibiyootigga iyadoo la adeegsanayo ensaymada bakteeriyada, taasoo kordhinaysa baaxadda dhaqdhaqaaqa iyo hagaajinta natiijooyinka daaweynta. Potassium clavulanate waxaa badanaa loo isticmaalaa isku-darka alaabada antibiyootigyada sida amoxicillin si loogu daaweeyo noocyo kala duwan oo caabuqyada bakteeriyada ah.
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Retapamulin CAS:224452-66-8
Retapamulin waa daawo antibiyootiko ah oo jirka la mariyo oo ka tirsan fasalka dawooyinka pleuromutilin. Waxaa loo isticmaalaa daaweynta caabuqyada maqaarka ee bakteeriyada, gaar ahaan impetigo oo ay keenaan noocyada nugul ee Staphylococcus aureus iyo Streptococcus pyogenes. Retapamulin wuxuu u shaqeeyaa isagoo joojinaya isku-darka borotiinka bakteeriyada, taasoo horseedaysa ciribtirka bakteeriyada cudurka qabta iyo xallinta caabuqa maqaarka.
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Staurosporine, streptomyces staurosporeus CAS:62996-74-1
Staurosporine waa badeeco dabiici ah oo laga soocay bakteeriyada Streptomyces staurosporeus. Waxaa loo kala saaraa inay tahay alkaloid awood leh oo leh dhaqdhaqaaq bayooloji oo muhiim ah, gaar ahaan ka hortagga kinase-ka borotiinka iyo kicinta apoptosis-ka unugyada. Staurosporine si ballaaran ayaa loo bartay sifooyinka daawada, oo ay ku jiraan awooddeeda ka hortagga kansarka iyo doorkeeda qalab cilmi baaris ah oo ku saabsan daraasadaha calaamadaynta unugyada.
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Cusbo disodium ah oo fosfoomycin ah CAS:26016-99-9
Cusbada disodium ee Phosphomycin waa antibiyootig ballaaran oo loo isticmaalo daaweynta caabuqyada bakteeriyada kala duwan. Waxay ka tirsan tahay fasalka asiidhyada fosfonic waxayna ka shaqeysaa joojinta sameynta derbiga unugyada bakteeriyada. Budadan crystalline-ka cad aad bay u milmaysaa biyaha waxaana badanaa lagu qaataa xidid ama afka. Cusbada disodium ee Phosphomycin waxaa loo yaqaanaa waxtarkeeda ka dhanka ah noocyo badan oo bakteeriya ah oo garaam-positive ah iyo garaam-negative ah, taasoo ka dhigaysa doorasho badan oo lagu daaweyn karo caabuqyada.
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Phleomycin CAS:11006-33-0
Phleomycin waa antibiyootig xooggan oo loo isticmaalo cilmi-baarista bayoolajiga molecular-ka si loo doorto unugyada ka kooban hiddo-wadaha xiisaha leh. Iyada oo leh farsamo ficil oo ku lug leh kala-goynta DNA-da, Phleomycin waxay waxtar u leedahay bakteeriyado kala duwan waxaana si weyn loogu isticmaalay codsiyada cilmi-baarista kala duwan. Antibiyootigan waxaa badanaa loo isticmaalaa iyadoo lala kaashanayo calaamadaha kale ee xulashada si loo abuuro khadadka unugyada deggan oo leh wax-ka-beddelka hidde-sidaha ee la doonayo. Phleomycin waxaa laga heli karaa labadaba dareere iyo budo, taasoo ka dhigaysa mid la isticmaali karo oo ku habboon dejinta tijaabada ee kala duwan. Cilmi-baarayaashu waxay qadarinayaan hufnaanteeda sare iyo isku halaynta ay ku leedahay xulashada unugyada la beddelay, taasoo ka dhigaysa qalab qiimo leh oo ku jira daraasadaha injineernimada hidde-sidaha.
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Penicillin V cusbo potassium ah CAS:132-98-9
Cusbada potassium-ka ee Penicillin V waa antibiyootiko afka laga qaato oo lagu daweeyo caabuqyada bakteeriyada. Waxa ku jira penicillin V, oo ah qaabka cusbada potassium-ka ee phenoxymethylpenicillin. Penicillin V waxay ka shaqeysaa faragelinta isku-darka peptidoglycan ee derbiga unugyada bakteeriyada. Tani waxay daciifisaa derbiga unugyada waxayna dishaa ama ka hortagtaa koritaanka bakteeriyada u nugul. Waxa loo heli karaa kiniinno ama dawooyin afka laga qaato si loogu daweeyo bukaan-socodka ee caabuqyada fudud ilaa kuwa dhexdhexaadka ah.
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Cusbo soodhiyam oo Penicillin G ah (cusbo soodhiyam oo Benzylpenicillin ah) CAS:69-57-8
Cusbada soodhiyamka ee Penicillin G waa antibiyootiko ka kooban penicillin G oo qaabkeeda cusbada soodhiyamka ah. Waxay ka shaqeysaa joojinta isku-darka lakabyada peptidoglycan ee derbiyada unugyada bakteeriyada, iyadoo disha bakteeriyada u nugul. Cusbada soodhiyamka ee Penicillin G waxaa laga heli karaa kiristaalo cad ama ku dhawaad cad oo ay tahay in loo beddelo xal ka hor duritaanka. Waxay bixisaa gaarsiin nidaamsan oo penicillin G ah si loogu daaweeyo caabuqyada bakteeriyada.
