-
N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea CAS:796848-79-8
N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea waa isku-dhis kiimiko ah oo leh qaacidada molecular-ka C10H11ClN2O2. Waxay ka tirsan tahay fasalka ka soo jeeda urea ee lagu beddelay kooxda chloro-hydroxyphenyl iyo kooxda cyclopropyl. Isku-darkaan waxaa loo aqoonsaday kakanaanta qaab-dhismeedka iyo codsiyada suurtagalka ah ee daraasadaha kiimikada iyo bayoolojiga ee kala duwan.
-
1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester CAS:205448-65-3
1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester waa isku-dhis kiimiko ah oo leh qaacidada molecular-ka C12H11NO4. Waxay ka tirsan tahay fasalka quinoline ee isku-dhisyada waxaana lagu gartaa koox methyl ester ah oo ku xiran giraanta quinoline, oo leh methoxy beddelka booska 7 iyo kooxda keto booska 4.
-
AZD-9291 mesylate CAS:1421373-66-1
AZD-9291 mesylate waa isku-dhis dawooyin ah oo leh qaacidada molecular-ka C28H33N7O4∙CH4O3S. Waxay ka tirsan tahay fasalka daawooyinka tyrosine kinase inhibitors waxaana inta badan loo isticmaalaa daaweynta kansarka sambabada unugyada aan yarayn (NSCLC). Daawadani waxay si gaar ah u bartilmaameedsataa oo u xakameysaa qaababka isbeddelay ee soo-dhoweeyaha koritaanka epidermal (EGFR), kuwaas oo badanaa laga helo burooyinka NSCLC.
-
5-Chloromethyl-2H-1,2,4-triazolin-3-one CAS:252742-72-6
5-Chloromethyl-2H-1,2,4-triazolin-3-one waa isku-dhis kiimiko oo muhiim ah oo leh codsiyo badan oo ku saabsan kiimikada daawada iyo cilmi-baarista beeraha. Waxay ka tirsan tahay fasalka ka soo jeeda triazolinone, oo lagu kala saaro qaab-dhismeed molecular oo gaar ah oo gacan ka geysta hawlaheeda bayoolojiga iyo isticmaalka daaweynta ee suurtagalka ah.
-
5-CHLOROTHIOPHEN-2-CARBONYL KLORIDE CAS:42518-98-9
5-Chlorothiophene-2-carbonyl chloride waa isku-dhis kiimiko ah oo ka tirsan fasalka thienylacyl chlorides. Waxaa lagu gartaa qaab-dhismeedkeeda molecular-ka oo ka kooban giraan thiophene ah oo lagu beddelay kooxda chloro ee booska 5-aad iyo kooxda carbonyl chloride ee booska 2-aad. Isku-darkani wuxuu xiiso weyn u leeyahay isku-darka dabiiciga ah sababtoo ah falcelintiisa kala duwan iyo codsiyada suurtagalka ah ee sayniska dawooyinka iyo agabka.
-
5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone CAS:503615-03-0
5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone waa isku-dhis kiimiko ah oo loo aqoonsaday qaab-dhismeedkeeda molecular-ka ee adag iyo codsiyada kala duwan ee kiimikada daawada iyo cilmi-baarista dawooyinka. Isku-darkani wuxuu ka tirsan yahay fasalka pyridinones waxaana lagu kala soocaa hab-raaciisa gaarka ah ee kooxaha shaqeynaya, kuwaas oo bixiya sifooyin gaar ah oo muhiim u ah hawlihiisa bayoolojiga.
-
4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester CAS:5909-24-0
4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester waa isku-dhis kiimiko ah oo loo aqoonsaday doorkeeda muhiimka ah ee kiimikada daawada iyo cilmi-baarista dawooyinka. Iyada oo ka tirsan qaybta ka soo jeeda pyrimidine, isku-darkani wuxuu muujinayaa qaab-dhismeed molecular oo gaar ah oo muhiim u ah hawlihiisa bayoolojiga iyo codsiyada daaweynta.
-
-
3-CHLORO-4-METHOXYBENZYLAMINE HYDROCHLORIDE CAS:41965-95-1
3-Chloro-4-Methoxybenzylamine Hydrochloride waa kiimiko caan ah oo si weyn loogu aqoonsaday isticmaalka kiimikada daawada iyo cilmi-baarista dawooyinka. Isku-darkani wuxuu ku jiraa fasalka amiinada udgoonka leh waxaana lagu kala soocaa hab-raaciisa gaarka ah ee kooxaha shaqeynaya ee muhiimka u ah hawlihiisa bayoolojiga.
-
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one CAS:545445-44-1
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one waa isku-dhis kiimiko ah oo caan ku ah qaab-dhismeedkeeda molecular-ka ee adag iyo codsiyada kala duwan ee kiimikada daawada iyo horumarinta daawada. Isku-darkani wuxuu ka tirsan yahay fasalka dihydropyridinones waxaana lagu gartaa isku-dubaridkiisa adag ee kooxaha shaqeynaya, kuwaas oo bixiya sifooyin gaar ah oo muhiim u ah hawlihiisa bayoolojiga.
-
L(-)-Aashitada Thiazolidine-4-karboxylic CAS:34592-47-7
L(-)-Thiazolidine-4-carboxylic acid waa isku-dhis kiimiko oo caan ah oo loo aqoonsaday adeegsigeeda kala duwan ee kiimikada daawada iyo cilmi-baarista dawooyinka. Iyada oo ka tirsan nooca thiazolidine derivatives, isku-darkani wuxuu leeyahay qaab-dhismeed molecular oo gaar ah oo muhiim u ah hawlihiisa bayoolojiga iyo kartida daaweynta.
-
Nintedanib CAS:656247-17-5
Nintedanib waa molecule yar oo awood leh oo tyrosine kinase inhibitor ah (TKI) oo leh muhiimad daaweyn oo muhiim ah oo ku saabsan cudurrada kansarka iyo fibrotic. Waxay ku lug leedahay saameynteeda daawooyinka iyadoo bartilmaameedsanaysa kinases badan oo tyrosine receptor ah oo ku lug leh angiogenesis, fibrogenesis, iyo nidaaminta koritaanka burooyinka.
