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Sitagliptin Phosphate CAS:654671-78-0 Alaab-qeybiye Soo-saare

Sitagliptin Phosphatewaa daawada ugu horreysa ee cusub ee dipeptidyl peptidase IV ee ka timaadda Merck si loogu daaweeyo nooca 2aad ee sonkorowga iyada oo aan la kordhin miisaanka, heerka hypoglycemia-na wuxuu la mid ahaa placebo. Sitagliptin wuxuu u shaqeeyaa isagoo kor u qaadaya nidaamka incretin ee jirka, kaas oo ka caawiya inuu nidaamiyo gulukooska isagoo saameeya unugyada β iyo α ee ganaca.


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Codsiga iyo Saamaynta

Sitagliptin Phosphate waa daawada trizolopyrazine dipeptidyl peptidase IV inhibitor. Sitagliptin dhawaan ayaa loo ansixiyay daaweynta nooca II ee sonkorowga. Sitagliptin phosphate waa daawada dipeptidyl peptidase Ⅳ (DDP-4) ee ay soo saartay shirkadda Jarmalka ee Merck waxayna markii ugu horreysay heshay oggolaanshaha Maamulka Cuntada iyo Dawooyinka ee Mareykanka si loogu daaweeyo nooca 2aad ee sonkorowga, waa daawo cusub oo ka hortagta sonkorowga, waxay hagaajin kartaa awoodda jirka ee uu ku yarayn karo heerarka sare ee gulukooska dhiigga, iyo incretin-ka dabiiciga ah ee sii kordhaya iyadoo la joojinayo dhaqdhaqaaqa enzyme-kan, oo ay ku jiraan heerarka glucagon-like peptide 1 iyo insulinotropic peptide-ka ku tiirsan gulukooska, taasoo kicinaysa ganaca inuu hagaajiyo wax soo saarka insulin oo uu joojiyo wax soo saarka gulukooska ee beerka, ugu dambayntiina uu yareeyo saameynta caafimaad ee fiirsashada gulukooska dhiigga.

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Macluumaad Dheeraad ah:

Halabuurka C16H15F6N5O.H3PO4
Baaritaan 99%
Muuqaalka Budada cad ilaa budo cad
Lambarka CAS. 654671-78-0
Baakad 25KG
Muddada Khafiska 2 sano
Kaydinta Ku kaydi meel qabow oo qalalan
Shahaadada ISO.

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