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Tetracycline CAS:60-54-8
Tetracycline waa antibiyootig ballaaran oo ka tirsan fasalka tetracycline, oo laga soo qaatay isku-darka dabiiciga ah ee chlortetracycline. Waxay joojisaa isku-darka borotiinka bakteeriyada iyadoo ku xidhan ribosome-ka bakteeriyada, taasoo ka hortagaysa ku-xidhka aminoacyl-tRNA ee isku-dhafka mRNA-ribosome. Habkan ficilku wuxuu horseedaa saameyn bacteriostatic ah oo ka dhan ah noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah, iyo sidoo kale protozoa gaar ah.
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Teicoplanin CAS:61036-62-2
Teicoplanin waa antibiyootiko glycopeptide ah oo laga soo qaatay Actinoplanes teichomyceticus, oo wax ku ool ah oo ka dhan ah bakteeriyada gram-positive kala duwan oo ay ku jiraan methicillin-resistant Staphylococcus aureus (MRSA). Waxay joojisaa isku-darka derbiga unugyada bakteeriyada iyadoo ku xidha terminus-ka D-alanyl-D-alanine ee horudhaca peptidoglycan, taasoo horseedaysa lysis unug iyo saameyn bakteeriya. Teicoplanin waxaa badanaa loo isticmaalaa goobaha caafimaadka si loogu daaweeyo caabuqyada daran ee ay keenaan noolaha gram-positive.
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Sulfisoxazol (4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide) CAS:127-69-5
Sulfisoxazole, oo sidoo kale loo yaqaan sulfifurazole, waa antibiyootig sulfonamide ah oo ka tirsan fasalka daawada sulfa. Si kiimiko ah ayaa loogu tilmaamay 4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide, sulfisoxazole wuxuu joojiyaa koritaanka bakteeriyada isagoo faragelinaya isku-darka folic acid. Habkan ficilku wuxuu bartilmaameedsadaa dihydropteroate synthase, oo ah ensaym muhiim u ah soo saarista bakteeriyada folate, taasoo carqaladeynaysa korriinkooda iyo fiditaankooda.
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Sulfapyridine CAS:144-83-2
Sulfapyridine waa antibiyootig sulfonamide ah oo taariikh ahaan loo isticmaali jiray daaweynta caabuqyada bakteeriyada, gaar ahaan intii lagu jiray Dagaalkii Labaad ee Adduunka. Waxay ka tirsan tahay nooca daawooyinka sulfa, kuwaas oo joojiya koritaanka bakteeriyada iyagoo faragelinaya isku-darka folic acid. Sulfapyridine waxay isticmaasha saameynteeda bakteeriyada iyadoo bartilmaameedsanaysa dihydropteroate synthase, oo ah ensaym muhiim u ah soo saarista folate ee bakteeriyada.
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Tazobactam CAS:89786-04-9
Tazobactam waa daawo ka hortagta beta-lactamase oo kor u qaadaysa firfircoonida antibiyootikada beta-lactam iyadoo ka ilaalinaysa burburka enzymes-ka beta-lactamase ee ay soo saaraan bakteeriyado badan oo iska caabiya. Waxaa si caadi ah loo isticmaalaa iyadoo lala kaashanayo antibiyootikada beta-lactam sida piperacillin si loo ballaariyo firfircoonidooda ka dhanka ah noocyo kala duwan oo caabuqyada bakteeriyada ah. Tazobactam si wax ku ool ah ayuu u soo celiyaa waxtarka antibiyootikada beta-lactam ee ka dhanka ah bakteeriyada soo saarta beta-lactamase, gaar ahaan noolaha garaam-negative.
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Tigecycline CAS:220620-09-7
Tigecycline waa antibiyootig glycylcycline oo ballaaran oo joojiya isku-darka borotiinka bakteeriyada isagoo ku xidha qaybta hoose ee ribosomal-ka 30S, taasoo keenta saameyn bakteeriya oo ka dhan ah noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah, oo ay ku jiraan jeermisyada daawada badan u adkaysta. Waxay si qaabaysan ula xiriirtaa tetracyclines laakiin waxay leedahay firfircooni la xoojiyay oo ka dhan ah noocyada iska caabbinta sababtoo ah farsamo gaar ah oo ficil iyo wax ka beddelka qaab-dhismeedka.
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Cusbo soodhiyam Sulbactam CAS:69388-84-7
Cusbada soodhiyamka Sulbactam waa daawo ka hortagta beta-lactamase oo si caadi ah loogu isticmaalo iyadoo lala kaashanayo antibiyootiko gaar ah si loola dagaallamo caabuqyada bakteeriyada. Waxay ka hortagtaa dhaqdhaqaaqa ensaymada beta-lactamase ee ay soo saarto bakteeriyada, kuwaas oo ka dhigi kara antibiyootiko kuwo aan waxtar lahayn. Iyadoo laga hortagayo burburka antibiyootigyada sida penicillins iyo cephalosporins, milixda soodhiyamka sulbactam waxay ka caawisaa inay kor u qaaddo sifooyinkeeda bakteeriyada dila. Isku-darkaan waxaa badanaa loo isticmaalaa iyadoo lala kaashanayo antibiyootiko sida ampicillin si loo abuuro saameyn isku-dhafan oo ka dhan ah noocyo badan oo bakteeriya ah oo u nugul.
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Sulfadimidine CAS:57-68-1
Sulfadimidine, oo sidoo kale loo yaqaan sulfamethazine, waa antibiyootig sulfonamide ah oo loo isticmaalo daaweynta caabuqyada bakteeriyada. Waxay ka tirsan tahay fasalka daawooyinka lidka ku ah jeermiska ee loo yaqaan daawooyinka sulfa, kuwaas oo ka shaqeeya joojinta koritaanka iyo taranka bakteeriyada. Sulfadimidine waxay faragelisaa isku-darka folic acid ee bakteeriyada, oo ah qayb muhiim u ah badbaadadooda, taasoo horseedaysa saameyn bakteeriya oo ka dhan ah noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah.
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Cusbo soodhiyam Sulfacetamide CAS:6209-17-2
Cusbada soodhiyamka ee Sulfacetamide waa nooc ka mid ah daawada sulfacetamide oo biyo ku milma, oo ah antibiyootiko sulfonamide ah oo si caadi ah loogu isticmaalo qaacidooyinka maqaarka lagu mariyo si loogu daaweeyo caabuqyada bakteeriyada ee maqaarka iyo indhaha. Qaabkan milixda ah wuxuu xoojiyaa milmida iyo xasilloonida sulfacetamide, taasoo ka dhigaysa mid ku habboon codsiyada dawooyinka kala duwan. Cusbada soodhiyamka ee Sulfacetamide waxay ka shaqeysaa joojinta koritaanka bakteeriyada, gaar ahaan kuwa mas'uulka ka ah xaaladaha sida finanka vulgaris, seborrheic dermatitis, iyo caabuqyada indhaha sida conjunctivitis. Waxay faragelisaa isku-darka bakteeriyada folate, iyadoo si wax ku ool ah u bartilmaameedsanaysa noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah.
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Streptomycin sulfate CAS:3810-74-0
Streptomycin sulfate waa daawo antibiyootiko ah oo ka tirsan fasalka aminoglycoside. Waxaa laga soo qaatay bakteeriyada Streptomyces griseus waxaana badanaa loo isticmaalaa in lagu daaweeyo caabuqyada bakteeriyada. Streptomycin sulfate wuxuu u shaqeeyaa isagoo joojinaya isku-darka borotiinka bakteeriyada, taasoo si wax ku ool ah u disha bakteeriyada nugul. Badanaa waxaa loo qoraa daaweynta qaaxada, cudurka daacuunka, tularemia, iyo caabuqyo kale oo gaar ah oo ay keento bakteeriyada nugul. Streptomycin sulfate badanaa waxaa lagu heli karaa qaab la isku duro waxaana lagu qaataa gudaha ama xididka iyadoo la kormeerayo caafimaadka.
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Cusbo soodhiyam Sulfamethoxazole CAS:4563-84-2
Cusbada soodhiyamka ee Sulfamethoxazole waa nooc ka mid ah bakteeriyada biyaha ku milma ee sulfamethoxazole, oo ah antibiyootiko sulfonamide ah oo loo isticmaalo daaweynta caabuqyada bakteeriyada. Qaabkan milixda ah wuxuu xoojiyaa milmida iyo xasilloonida sulfamethoxazole, taasoo ka dhigaysa mid ku habboon qaacidooyinka dawooyinka kala duwan. Cusbada soodhiyamka ee Sulfamethoxazole waxay samaysaa saameynteeda bakteeriyada iyadoo joojinaysa isku-darka folic acid ee bakteeriyada, taasoo ah hab lagama maarmaan u ah korriinkooda iyo tarmintooda. Waxay waxtar u leedahay noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah.
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Sulfamethoxazole CAS:723-46-6
Sulfamethoxazole waa antibiyootig sulfonamide ah oo si caadi ah loo isticmaalo iyadoo lala kaashanayo trimethoprim si loo sameeyo daawo awood leh oo bakteeriyada disha oo loo yaqaan co-trimoxazole ama trimethoprim-sulfamethoxazole (TMP-SMX). Waxay ka tirsan tahay fasalka daawooyinka lidka ku ah bakteeriyada ee loo yaqaan daawooyinka sulfa, kuwaas oo joojiya koritaanka bakteeriyada iyagoo faragelinaya isku-darka folic acid. Sulfamethoxazole si gaar ah ayuu u bartilmaameedsadaa dihydropteroate synthase, oo ah ensaym ku lug leh soo saarista folate, sidaas darteedna wuxuu sameeyaa saameyn bacteriostatic ah oo ka dhan ah noocyo badan oo bakteeriya garaam-positive ah iyo garaam-negative ah.
