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Ezetimibe INT A CAS:189028-95-3
Ezetimibe INT A waa isku-darka dawooyinka loogu talagalay in lagu daaweeyo hyperlipidemia, oo lagu garto heerarka kolestaroolka oo sarreeya. Waxay joojisaa nuugista xiidmaha ee kolestaroolka iyo sterol-yada la xiriira iyadoo bartilmaameedsaneysa borotiinka Niemann-Pick C1-like 1 (NPC1L1), taasoo hoos u dhigaysa heerarka guud ee kolestaroolka dhiigga.
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Pramipexole CAS:104632-26-0
Pramipexole waa daawo dopamine agonist ah oo loo isticmaalo daaweynta cudurka Parkinson iyo xanuunka lugaha aan nasashada lahayn (RLS). Waxay ka shaqeysaa kicinta soo-dhoweeyayaasha dopamine ee maskaxda, taasoo hagaajinaysa calaamadaha dhaqdhaqaaqa ee cudurka Parkinson iyo yareynta dareenka aan raaxada lahayn ee RLS. Pramipexole waxaa laga heli karaa labadaba daawooyinka si degdeg ah loo sii daayo iyo kuwa sii daaya ee dheeraadka ah, iyadoo bixisa dabacsanaan ku saabsan fursadaha daaweynta ee bukaanada.
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R-Tetrahydropapaverine hydrochloride CAS:54417-53-7
R-Tetrahydropapaverinehydrochloride waa kiimiko asal ahaan loo isticmaalo cilmi-baarista dawooyinka. Waxaa loo yaqaanaa isticmaalka suurtagalka ah ee horumarinta daawooyinka lagu bartilmaameedsanayo xanuunnada neerfaha iyo wadnaha iyo xididdada dhiigga. Isku-darkaan waxaa loo sameeyay oo lagu bartay sifooyinka daawada, gaar ahaan saameynta uu ku leeyahay muruqyada siman ee xididdada dhiigga iyo nidaamyada neerfaha. Cilmi-baarayaashu waxay baaraan saameyntiisa daaweynta ee suurtagalka ah ee xaaladaha sida dhiigkarka iyo xaaladaha neerfaha qaarkood, iyagoo ujeedadoodu tahay inay u adeegsadaan astaamaha daawada ee codsiyada caafimaad ee mustaqbalka.
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4-(4-Aminophenyl)morpholin-3-one CAS:438056-69-0
4-(4-Aminophenyl)morpholin-3-one waa isku-dhis kiimiko ah oo leh qaacidada molecular-ka C11H14N2O2. Waxaa sidoo kale loo yaqaanaa magaca IUPAC, 4-(4-Aminophenyl)morpholin-3-one. Isku-darkani wuxuu leeyahay giraan morpholine ah oo lagu beddelay koox aminophenyl ah oo ku taal booska 4-aad.
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3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone CAS:272778-12-8
3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone waa isku-dhis kiimiko oo isku dhafan oo leh qaacidada molecular-ka C34H41F2N3O6Si2. Waa nooc ka mid ah oxazolidinone oo loo yaqaan kakanaanta qaab-dhismeedka iyo codsiyada dawooyinka ee suurtagalka ah.
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4-hydroxythiobenzamide CAS:25984-63-8
4-Hydroxythiobenzamide waa isku-dhis kiimiko ah oo loo yaqaan qaab-dhismeedkeeda oo leh koox hydroxy ah oo ku xiran xudunta thiobenzamide. Waxaa loo isticmaalaa isku-darka dabiiciga ah iyo cilmi-baarista kiimikada sababtoo ah sifooyinka shaqo ee gaarka ah iyo codsiyada suurtagalka ah ee qaybaha kala duwan ee sayniska.
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(S)-4,5,6,7-Tetrahydro-2,6-benzothiazolediamine CAS:106092-09-5
(S)-4,5,6,7-Tetrahydro-2,6-benzothiazolediamine waa isku-dhis kiimiko ah oo loo aqoonsaday qaab-dhismeedkeeda oo leh xudunta benzothiazole iyo kooxda amine ee shaqaynaysa. Waxaa lagu bartaa isticmaalka suurtagalka ah ee cilmi-baarista dawooyinka iyo isku-darka dabiiciga ah, sababtoo ah qaab-dhismeedkeeda gaarka ah ee molecular-ka.
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Bupivacaine CAS:2180-92-9
Bupivacaine waa suuxdin maxalli ah oo muddo dheer shaqeyneysa oo ka tirsan fasalka daawooyinka amide. Waxay ka shaqeysaa iyadoo xannibaysa calaamadaha neerfaha ee jirka, taasoo keenta kabuubyo ama luminta dareenka meel gaar ah. Bupivacaine waxaa badanaa loo isticmaalaa yareynta xanuunka inta lagu jiro qalliinka, dhalmada, iyo waxqabadyada kale ee caafimaadka. Waxaa sidoo kale loo isticmaalaa maaraynta xanuunka qalliinka ka dib iyo xaaladaha qaarkood ee xanuunka daba dheeraada. Bupivacaine waxaa lagu duraa irbad waxaana loo yaqaanaa saameynteeda xooggan iyo tan waarta ee bixinta xanuunka.
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Atracurium oxalate CAS:64228-78-0
Atracurium oxalate waa isku-darka daawada loo isticmaalo sidii wakiilka xanniba muruqyada neerfaha ee suuxinta. Waa nooc ka mid ah atracurium besylate, oo loogu talagalay in lagu maamulo xididada inta lagu jiro qalliinka si loo kiciyo nasashada murqaha. Isku-darkani wuxuu u shaqeeyaa si tartan ah isagoo ku xidha qabtayaasha cholinergic ee isgoyska neerfaha, taasoo joojinaysa gudbinta dareenka neerfaha waxayna keentaa curyaannimo ku meel gaar ah oo muruqyada lafaha ah. Atracurium oxalate waxaa lagu qiimeeyaa bilawga degdega ah iyo muddada dhexdhexaadka ah ee ficilka, taasoo ka dhigaysa mid ku habboon hababka qalliinka ee kala duwan ee u baahan nasashada murqaha la xakameeyey.
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Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate CAS:161797-99-5
Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate waa isku-dhis kiimiko ah oo loo adeegsado cilmi-baarista dawooyinka iyo isku-darka dabiiciga ah. Waxay ka tirsan tahay qoyska thiazole waxaana lagu gartaa kooxaha phenyl iyo ester ee la beddelay. Isku-darkaan waxaa lagu bartaa hawlihiisa bayoolojiga ee suurtagalka ah waxaana loo sameeyay ujeeddooyin cilmi-baaris oo kala duwan oo ku saabsan kiimikada daawada.
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2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole CAS:104617-49-4
2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole waa isku-dhis kiimiko ah oo loo yaqaan qaab-dhismeedkeeda oo leh xudunta benzothiazole iyo laba kooxood oo amino ah. Waxaa loo aqoonsan yahay codsigeeda suurtagalka ah ee cilmi-baarista dawooyinka iyo isku-darka dabiiciga ah, sababtoo ah qaab-dhismeedkeeda gaarka ah ee molecular-ka.
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4-[[(4-Fluorophenyl)imino]methyl]-phenol CAS:3382-63-6
4-[[(4-Fluorophenyl)imino]methyl]-phenol, oo leh qaacidada molecular-ka C13H10FNO, waa isku-dhis kiimiko ah oo loo yaqaan qaab-dhismeedkeeda udgoon. Waxay leedahay giraan phenol ah oo lagu beddelay koox iminomethyl ah oo ku xiran qayb fluorophenyl ah.
